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Cat No. | Product Name | Synonyms | Targets |
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T22381 | Antimalarial agent 14 | 4-hydroxy-3-phenyl-naphthalene-1,2-dione,2-Hydroxy-3-phenyl-1,4-naphthoquinone | Others |
Antimalarial agent 14 (NSC-102533) is a bioactive chemical. | |||
T25621 | Lankacidinol A | Lankacidinol 14-acetate,Antibiotic T-2636D,P 2636 D,P2636 D,P-2636 D | |
Lankacidinol A is a metabolite of macrolide antibiotic. | |||
T40344 | CBP/p300-IN-14 | CBP/p300-IN-14 | |
CBP/p300-IN-14, efficiently inhibits CBP/EP300 (lysine acetyltransferase) with an IC50 value of 3.3 nM. | |||
T34734 | Substance P (1-4) | SP(1-4) | |
Substance P (1-4) is a substance P N-terminal tetrapeptide fragment. | |||
T0120 | Voriconazole | UK-109496 | Antifection , Antifungal |
Voriconazole (UK-109496) is a triazole antifungal agent that specifically inhibits STEROL 14-ALPHA-DEMETHYLASE and CYTOCHROME P-450 CYP3A. | |||
T6686 | Sulconazole mononitrate | Exelderm,Sulconazole Nitrate,RS 44872 | Antibacterial , Antibiotic , Antifungal |
Sulconazole mononitrate (Exelderm) is the nitrate salt form of sulconazole, a synthetic imidazole derivative with the antifungal property. Sulconazole mononitrate inhibits fungal cytochrome P-450 sterol C-14 alpha-demeth... | |||
T36949 | Niaprazine | 5-HT Receptor , Adrenergic Receptor , Histamine Receptor | |
Niaprazine is a histamine H1-receptor antagonist with marked sedative properties. Niaprazine has antihistamine and antiserotonin activities and can be used for sleep disorder research[1][2]. Niaprazine exhibits a low aff... | |||
T25591 | Lab 170250F | Lab-170250F,Lab170250F | |
Lab 170250F is a potent cytochrome P-450-obtusifoliol-14-demethylase inhibitor. | |||
T69167 | Buthiobate | ||
Buthiobate is a fungicide which inhibits lanosterol 14 alpha-demethylation catalyzed by a cytochrome P-450. | |||
T37025 | Mca-PLAC(p-OMeBz)-WAR(Dpa)-NH2 | Mca-PLAC(p-OMeBz)-WAR(Dpa)-NH2 | |
Mca-PLAC(p-OMeBz)-WAR(Dpa)-NH2 is a fluorogenic substrate for matrix metalloproteinase-14 (MMP-14). Upon cleavage by MMP-14, 7-methoxycoumarin-4-acetyl (Mca) is released and its fluorescence can be used to quantify MMP a... | |||
T63235 | KRAS inhibitor-14 | ||
KRAS inhibitor-14 is a potent inhibitor of KRAS G12C (IC50: 0.249 μM). KRAS inhibitor-14 exhibited p-ERK inhibition in MIA PaCA-2, A549 cells with IC50s of 1.12, >33.3 μM, respectively. KRAS inhibitor-14 has potential to... | |||
T63887 | SOS1-IN-14 | ||
SOS1-IN-14 is a selective, potent, orally active SOS1 inhibitor (IC50: 3.9 nM). sOS1-IN-14 is absorbed in the intestine using a P-glycoprotein-mediated efflux mechanism. sOS1-IN-14 can be used in the study of KRAS mutate... | |||
T73310 | AXL-IN-14 | TAM Receptor | |
AXL-IN-14 is a potent, orally active inhibitor of AXL with an IC50 of 0.8 nM that effectively suppresses Gas6/AXL-mediated cell migration and invasion, reduces the expression of p-AXL and p-AKT proteins, and demonstrates... | |||
T75996 | Murepavadin TFA | ||
Murepavadin (POL7080) (TFA), a 14-amino-acid cyclic peptide, serves as a highly potent, specific antibiotic with remarkable antimicrobial activity against P. aeruginosa, demonstrated by MIC 50 and MIC 90 values of 0.12 m... | |||
T37362 | 7α-Thiomethylspironolactone | ||
7α-Thiomethylspironolactone is a major metabolite of the synthetic steroid spironolactone.1,2 1.Jankowski, A., Skorek-Jankowska, A., and Lamparczyk, H.Simultaneous determination of spironolactone and its metabolites in h... | |||
T68581 | AP23464 | ||
AP23464 is a potent adenosine 5'-triphosphate (ATP)-based inhibitor of Src and Abl kinases, displays antiproliferative activity against a human CML cell line and Bcr-Abl-transduced Ba/F3 cells (IC(50) = 14 nM. AP23464 ab... | |||
T36470 | Biotinyl hexylamine | ||
Biotinyl hexylamine is a synthetic intermediate.1,2It has been used in the synthesis of avidin nucleic acid nano assemblies (ANANAS) and chemotherapeutic conjugates for the diagnosis of, and drug delivery to, tumors. 1.S... | |||
T36152 | 14S(15R)-EET | ||
14S(15R)-EET is an oxylipin and a cytochrome P450 metabolite of arachidonic acid .114S(15R)-EET binds to isolated guinea pig monocytes with a Kivalue of 612.5 nM in a competitive binding assay using [3H]14(15)-EET.2It in... | |||
T35463 | (±)14(15)-EET | (±)14,15-EET,(±)14,15-EpETrE,(±)14(15)-EET | |
(±)14(15)-EET is a metabolite of arachidonic acid that is formed via epoxidation of arachidonic acid by cytochrome P450.[1],[2] It prevents increases in leukotriene B4, ICAM-1, and chemokine (C-C motif) ligand 1 (CCL2) i... | |||
T37412 | AZ-GHS-22 | ||
AZ-GHS-22 is an inverse agonist of the growth hormone secretagogue receptor 1a (GHS-R1a), which is also known as the ghrelin receptor.1It binds to GHS-R1a with an IC50value of 0.77 nM. AZ-GHS-22 decreases food intake in ... | |||
T67442 | CGP-53716 | ||
The growth factors, platelet-derived growth factor (PDGF) and basic fibroblast growth factor (bFGF) play major roles in enhanced smooth muscle cells growth in rodent blood vessels after vascular injury. Tyrosine kinase i... | |||
T36108 | YW3-56 (hydrochloride) (technical grade) | YW3-56 (hydrochloride) (technical grade) | |
YW3-56 is an inhibitor of protein arginine deiminase 2 (PAD2) and PAD4 (IC50s = 0.5-1 and 1-5 μM, respectively).1It inhibits the growth of U2OS osteosarcoma cells (IC50= ~2.5 μM) in a p53-dependent mannerviainduction of ... | |||
T36296 | BIO5192 hydrate | ||
BIO5192 hydrate is a selective and potent integrin α4β1 (VLA-4) inhibitor (Kd<10 pM). BIO5192 hydrate selectively binds to α4β1 (IC50=1.8 nM) over a range of other integrins. BIO5192 hydrate results in a 30-fold increase... |
Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
TN3283 | 8alpha-Hydroxylabda-13(16),14-dien-19-yl p-hydroxycinnamate | Others | |
8alpha-Hydroxylabda-13(16),14-dien-19-yl p-hydroxycinnamate is a natural product for research related to life sciences. The catalog number is TN3283 and the CAS number is 117254-98-5. | |||
TN6121 | 4''-O-trans-p-Coumaroylafzelin | Kaempferol 3-O-(4''-O-trans-p-coumaroyl)rhamnopyranoside | |
4''-O-trans-p-Coumaroylafzelin is a natural product for research related to life sciences. The catalog number is TN6121 and the CAS number is 623927-14-0. | |||
T35624 | Ajoene | ||
Ajoene is a disulfide that has been found inA. sativumand has diverse biological activities, including antibacterial, anticancer, antiplatelet, and antioxidant properties.1,2,3,4It is active against Gram-positive (MICs =... |
Cat No. | Product Name | Species | Expression System |
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TMPY-01357 | S100A9 Protein, Human, Recombinant (His) | Human | Baculovirus Insect Cells |
S100A9 Protein, Human, Recombinant (His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 14.6 kDa and the accession number is P06702. | |||
TMPY-01330 | S100A9 Protein, Human, Recombinant | Human | E. coli |
S100A9 Protein, Human, Recombinant is expressed in E. coli expression system. The predicted molecular weight is 26 and 13 kDa and the accession number is P06702. | |||
TMPY-06693 | Cor a 14 Protein, Corylus avellana, Recombinant | Corylus avellana | P. pastoris (Yeast) |
Cor a 14 Protein, Corylus avellana, Recombinant is expressed in P. pastoris yeast expression system. The predicted molecular weight is 10.5 kDa. | |||
TMPY-01816 | Pentraxin 3 Protein, Human, Recombinant (His) | Human | HEK293 Cells |
Pentraxin-related protein PTX3, also known as Tumor necrosis factor alpha-induced protein 5, Tumor necrosis factor-inducible gene 14 protein, TSG-14, PTX3 and TNFAIP5, is a secreted protein that contains one pentaxin dom... |